[PDF] Top 20 Design and synthesis of pironetin analogue/combretastatin A 4 hybrids containing a 1,2,3 triazole ring and evaluation of their cytotoxic activity
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Design and synthesis of pironetin analogue/combretastatin A 4 hybrids containing a 1,2,3 triazole ring and evaluation of their cytotoxic activity
... prepare cytotoxic TBMs with a dual ability to bind to either the a - or the b - tubulin subunits [19] and exert a microtubule-destabilizing ...by pironetin (binds to a -tubulin) and ... See full document
9
Design and Synthesis of Pironetin Analogue/Colchicine Hybrids and Study of Their Cytotoxic Activity and Mechanisms of Interaction with Tubulin
... Total synthesis of (−)-PA-48153C, a novel immunosuppressive 2- pyranone ...Total synthesis of a potent immunosuppressant ...Total synthesis of (−)-PA-48153C ... See full document
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TítuloInnovative three step microwave promoted synthesis of N propargyltetrahydroquinoline and 1,2,3 triazole derivatives as a potential factor Xa (FXa) inhibitors: drug design, synthesis, and biological evaluation
... management of thrombosis. In recent years, various pharmacological activities of N-heterocyclic compounds including tetrahydroquinoline (Figure 4d) have received immense importance because of ... See full document
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Design and Synthesis of Pironetin Analogue/Combretastatin A 4 Hybrids and Evaluation of Their Cytotoxic Activity
... structures and the observed cytotoxicity deserve comment. In the case of two subsets of hybrid molecules [27] where there are differences between in the carbon chain length ...(e.g. 1-4 ... See full document
18
SYNTHESIS OF GERANYLHYDROQUINONE DERIVATIVES WITH POTENCIAL CYTOTOXIC ACTIVITY
... concentration of the drug, required for 50% inhibition in vitro after 72 h of continuous exposure to the test ...µM) of each sample were evaluated in ...Table 1. The derivatives compounds ... See full document
10
Synthesis and cytotoxic activity of tri acyl ester derivatives of uridine in breast cancer cells
... Figure 2, shows the results of cell viability obtained by MTT assay with uridine, tri-esterified derivatives and ...uridine and its derivatives, to the lower concentrations evaluated, did not ... See full document
9
Synthesis and antiproliferative activity of new cyclodiprenyl phenols against select cancer cell lines
... compounds 2–5 had strong inhibitory effects on various cancer cell line growth and certain selectivity in relation to non-tumoral cells, we decided to study the effect of these ...compounds ... See full document
13
Design and Evaluation of a Scalable and Reconfigurable Multi Platform System for Acoustic Imaging
... family of devices from National Instruments that is oriented to sensors with nonstandard acquisition procedures, allowing low-level programming of the acquisition ...FPGA and a dual-core ARM ® ... See full document
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Synthesis and conformational analysis of leptocarpin derivatives Influence of modification of the oxirane ringon leptocarpin's cytotoxic activity
... transformation of Leptocarpin was obtained through the acid treatment of the leptocarpin with saturated chloroformic solution with HCl, to mimick what would happen when the drug encounters the gastric acid ... See full document
15
KNbO3 as Photocatalyst for Hydrogen Production
... g of each KN Photocatalyst was evaluated by splitting of the water molecule, using a 250W mercurial lamp and adding methanol to the water reactor system as sacrificial agent (2% ... See full document
8
(BIo)analytical microsystems based on the use of nanoparticles. Microreactors for the synthesis of nanoparticles
... molecules and their bulk ...focusing their investigations on this “new” technology in order to develop novel materials with unique and unusual ...fabrication of nanomaterials requires a ... See full document
329
Synthesis, Cytotoxic and Antimicrobial activities of 5-benzylidene-2- [(pyridine-2-ylmethylene)hydrazono]-thiazolidin-4-one Derivatives
... As complementary biological test, all 4-thiazolidinones were evaluated for antimicrobial activity against various bacterial and fungal species..[r] ... See full document
1
Antiplasmodial and Cytotoxic Activity of Piper Piedecuestanum Trel and Yunck
... species of Piper are economically important, among them Piper nigrum from which the pepper is obtained, condiment popularly used all over the ...range of traditional foods has been reported in the treatment ... See full document
9
Amidinate Aluminium Complexes as Catalysts for Carbon Dioxide Fixation into Cyclic Carbonates
... change of cocatalyst from tetrabutylam- monium bromide to tetrabutylammonium iodide has a positive effect for each of complexes 1–6, the conversion of styrene oxide 7a into styrene carbonate ... See full document
7
Platinum and palladium complexes with 2,4-Dinitrophenylhydrazine: synthesis and cytotoxic activity
... These complexes were characterized and the results shown that the ligand is coordinated to platinum or palladium by the basic nitrogen of NH 2 group and have the general structure cis- [r] ... See full document
1
Synthesis and cytotoxic activity of per acetylated and halogenated derivatives of nucleosides in breast cancer cells
... for 3’,4’,6’-O-acetyl-uridine in DMSO-d6 presents at high-field, a multiplet coupling with shift ...overlapping of H-5’ and H-6’ protons of ribose ring) with a high deshielding ... See full document
10
Hemi Synthesis and Anti Oomycete Activity of Analogues of Isocordoin
... efficient synthesis of a series of 4 0 -oxyalkyl-isocordoin analogues (2–8) is reported for the first ...time. Their structures were confirmed by 1 H-NMR, 13 C-NMR, ... See full document
9
Synthesis of Pyrrolidine Fused 1,3 Dithiolane Oligomers by the Cycloaddition of Polycyclic Dithiolethiones to Maleimides and Evaluation as Mercury(II) Indicators
... case of monoadducts 10, the presence of a maleimide 194 nucleus makes the products suitable for a second cycloaddition 195 ...7 and 2 equiv of 196 maleimide 10a reacted in re fl uxing ... See full document
14
Multivalent Molecular Shuttles – Effect of Increasing the Number of Centers in Switchable Catalysts
... in their structure have attracted the attention of many authors in this decade 1 demonstrating their suitability as an effective reaction ...developed 2 inspired by how nature can ... See full document
8
Desarrollo de dos nuevas sondas fluorogénicas derivadas de la bis-vainillina para la detección de catiónes metalicos trivalentes
... The design and synthesis of new chemosensors for the determination of metal cations represent an area of hight interest in supramolecular ...detection and cuantification ... See full document
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