[PDF] Top 20 Synthesis and Anti-HIV Activity Evaluation of 2-(5-(Naphthalen-1-yl)-1,2,3-thiadiazol-4-ylthio)-N-acetamides Derivatives
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Synthesis and Anti-HIV Activity Evaluation of 2-(5-(Naphthalen-1-yl)-1,2,3-thiadiazol-4-ylthio)-N-acetamides Derivatives
... development of novel HIV-1 non-nucleoside reverse transcriptase inhibitors (NNRTIs) offers the possibility of generating novel structures of increased ...novel ... See full document
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Design and synthesis of pironetin analogue/combretastatin A 4 hybrids containing a 1,2,3 triazole ring and evaluation of their cytotoxic activity
... (HT-29 and MCF-7) cell lines has then been measured. Several of the synthetic derivatives proved cytotoxic towards at least one of the two tumoral cell lines, with some of them showing ... See full document
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Synthesis and Multitarget Biological Profiling of a Novel Family of Rhein Derivatives As Disease Modifying Anti Alzheimer Agents
... form of the more lipophilic and cell permeable doubly acetylated prodrug ...Inhibition of A β 42 and Tau Aggregation in Intact Escherichia coli ...aggregation of two amyloidogenic ... See full document
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Design and Synthesis of Pironetin Analogue/Combretastatin A 4 Hybrids and Evaluation of Their Cytotoxic Activity
... measurement of the cytotoxicity of the synthetic combretastatin A-4 derivatives 1-4 and their enantiomers, 5-8, 9a-12a and ...ent-14 and 15 were also ...HT-29 and the ... See full document
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TítuloInnovative three step microwave promoted synthesis of N propargyltetrahydroquinoline and 1,2,3 triazole derivatives as a potential factor Xa (FXa) inhibitors: drug design, synthesis, and biological evaluation
... management of thrombosis. In recent years, various pharmacological activities of N-heterocyclic compounds including tetrahydroquinoline (Figure 4d) have received immense importance because of ... See full document
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Synthesis and antiproliferative activity of new cyclodiprenyl phenols against select cancer cell lines
... treatment of cancer ...avinosol and avarol offer promising opportunities for the development of new antitumor agents ...potential of meroterpenes is of great interest; however, low ... See full document
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Synthesis and evaluation of the antifungal activity of 2-(substituted-amino)-4,5-dialkyl-thiophene-3- carbonitrile derivatives
... All compounds presented fungicidal activity at different doses, but a few compounds showed moderate or poor antifungal activity when compared with the standard drugs. The Cryp- tococcus[r] ... See full document
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In vitro and in vivo evaluation of 2 aminoalkanol and 1,2 alkanediamine derivatives against Strongyloides venezuelensis
... nematodes of the genus Strongyloides, which are widely present in tropical and subtropical areas with climate suitable for the survival of larval stages of the species of this ... See full document
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TítuloANN multiscale model of anti HIV Drugs activity vs AIDS prevalence in the US at county level based on information indices of molecular graphs and social networks
... molecular and population ...types of input data coming from many different levels of organization of ...the anti-HIV drugs including at least the chemical structure of the ... See full document
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Synthesis and Release of Catecholamines by the Cat Carotid Body in Vitro: Effects of Hypoxic Stimulation
... (Biomedical Division).. synthesis, release, receptor localization, etc. ) with changes in chemoreceptor activity, and (2) the phar- macological characterization of the [r] ... See full document
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Comparative pharmacological evaluation of Hypericum perforatum and Rosmarinus officinalis for anti-depressant activity
... The herbal extracts of Hypericum perforatum (20 mg/kg/ p.o. ) were subjected for its antidepressant activity using four different animal models of depression, viz: Forced Swimming Test[r] ... See full document
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Desarrollo de dos nuevas sondas fluorogénicas derivadas de la bis-vainillina para la detección de catiónes metalicos trivalentes
... geometries of the molecules studied, with and without the cation were optimized and vibrational frequencies were calculated to ensure the validity of each ...global and FMO energies ... See full document
5
Synthesis and characterization of new alkoxide and aryloxide derivatives of titanium and zirconium X ray molecular structure of [ZrCp2(OC6F5)2]
... A clean reaction takes place when the ~-oxo compound [ZrCp2Mez/x-O] is treated with two equivalents of pentafluorophenol, leading to the isolation of the alkoxo complex [{ZrfP2Of6Fs}2/.t[r] ... See full document
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3. SAPOGENINS FROM THE HUSK OF CHENOPODIUM QUINOA, THE OBTAINING OF THEIR DERIVATIVES, AND THE EVALUATION OF THEIR CYTOTOXIC ACTIVITY.
... Cytotoxic evaluation The cytotoxicity of the four isolated sapogenins was evaluated in one normal-like human breast epithelial cell line MCF-10A and in one breast cancer cell line JIMT-1[r] ... See full document
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Synthesis, characterization, determination of luminescent properties of tetracoordinate organoboron compounds derivatives from organic tridentate ligands, and their potential application in OLEDs
... design and synthesis of new boron compounds, which has improved the chemical and optical properties in comparison to aluminum derivatives such as good solubility in organic solvents, ... See full document
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2. SYNTHESIS OF THE ANTI-CANCER CARBOPLATIN OXIDIZED, AND STUDY OF ITS INTERACTIONS WITH N-BASES BY CYCLIC VOLTAMMETRY.
... ocurrió en - 650 mV; también indicaron que el platino (IV) interacciona con el DNA con un solo enlace, como se puede ver en la figura 1c. Estos resultados se confirmaron por difracción de rayos X [7]. Un experimento in ... See full document
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Amidinate Aluminium Complexes as Catalysts for Carbon Dioxide Fixation into Cyclic Carbonates
... merisation of the epoxide took place without insertion of carbon dioxide under these reaction ...formation of cyclic carbonate 10 b in 80% isolated yield (Table 5, entry ...c and 10d were ... See full document
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2. EVALUATION OF FLAVONOID CONTENTS AND ANTIBACTERIAL ACTIVITY OF FIVE BOLIVIAN BACCHARIS SPECIES.
... Quantification of TFC Total Flavonoids Contents in the 5 Bolivian Baccharis expressed in mg of Luteolin equivalent per g of EtOH Extracts EE and Enriched Fraction by Sephadex LH-20 EFS..[r] ... See full document
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A new approach to the synthesis of 2 aminoimidazo[1,2 a]pyridine derivatives through microwave assisted N alkylation of 2 halopyridines
... Method B afforded 2e in a 55% yield the reaction mixture was stirred for 6 h at room temperature Mp 110-112 °C dec yellow powder, EtOAc.. Acknowledgements This research was supported by [r] ... See full document
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Evaluacin de resultados de VIH, ETS y CD4 en asistentes al programa de VIH/SIDA de la Ciudad de Mxico
... rapid HIV-antibody test, followed by Ag/Ab Combo HIV, HBsAg, anti-HVC and anti-TP CLIA testing applied in parallel to all ...fall of 2011, CD4 count and HIV-1 viral ... See full document
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