[PDF] Top 20 Soberanía alimentaria y el principio campesino
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The Docking Studies of New Derivatives of N-Phenylanthranilic Acids as Inhibitors of Microsomal Prostaglandin E Synthase-1 (mPGES-1)
... compound 25 , in which the hydrogen bonds are formed by carbonyl oxygen atoms of anthranilic acid 151. with Arg73 and Tyr117 in the molecule complex with mPGES-1[r] ... See full document
18
Docking Studies of the Derivatives of 3 oxamoyl(succinoyl)amides of N Phenylanthranilic Acids as Inhibitors of Enzymes COX 1 and COX 2
... Conducted docking studies found that pharmacological activity is associated with inhibiting prostaglandin synthesis by new derivatives of N-phenylanthranilic acid by ... See full document
80
SYNTHESIS, INSILICO DOCKING AND ADMET STUDIES OF ARYL ACETIC ACID DERIVATIVES AS PROSTAGLANDIN ENDOPEROXIDE H SYNTHASE 2 INHIBITORS
... the docking results are listed in Table ...the docking score, non-bonded interactions and Glide ...amino acids of 1PGE with iodosuprofen were Tyr 355, Arg120, Ser 530 and are shown in ... See full document
5
Linking microsomal prostaglandin E synthase-1/PGE-2 pathway with miR-15a and -186 expression: Novel mechanism of VEGF modulation in prostate cancer
... VEGF, mPGES-1, HIF-1α and Dicer, and for 30 min in TRIS buffer (pH 9) in a microwave at 500 W for ...of mPGES-1 (1:50, Thermo Scientific), VEGF (1:100, Merck Millipore), CD31 ... See full document
173
Studies of synthetic chalcone derivatives as potential inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and pro-inflammatory cytokines
... NP40 1%, NaCl 150 mM, EDTA 2 mM, Na 3 VO 4 200 mM, SDS ...Table 1 inhibition of secretory phospholipase a 2 -V (sPla 2 -V), cOX-1, cOX-2 and lOX-15 activities by synthetic chalcone ... See full document
7
Molecular Docking Study of Certain Plant Alkaloid Derivatives as Inhibitors of Various Drug Targets of Alzheimer’s Disease
... discover inhibitors with high binding capabilities with a protein target, drug- likeliness properties, and ADMET (Absorption, Distribution, Metabolism, Excretion, and Toxicity) ...of new compounds based ... See full document
15
Synthesis, antibacterial activity and molecular docking studies of N' benzylidene/N' (1 phenylethylidene)hexa 2,4 dienehydrazide derivativesf
... molecular docking of sorbic acid, ester and their hydrazides (1-11) was performed using ...present docking study Cys112 and Ala246 was found to be responsible for substrate binding and cleavage of ... See full document
61
MOLECULAR DOCKING STUDIES OF A FEW NOVEL PYRIMIDINE DERIVATIVES AS REVERSE TRANSCRIPTASE HIV 1 INHIBITORS
... Pyrimidine-based derivatives are studied for their HIV-1 reverse transcriptase inhibition activities using in-silico ...pyrimidine-based derivatives designed using computer-based molecule designed ... See full document
24
QSAR Studies of Lanosterol Synthase Inhibitors as Potential Antihypercholesterolemic Compounds
... QSAR study was performed on the data set consists of twenty three compounds having LSS inhibitory activity. The biological activity data IC 50 (nm) were changed to pIC 50 for QSAR analysis. The pIC 50 values of the ... See full document
26
Pharmacophore Modeling, Atom based 3D-QSAR and Docking Studies of Chalcone derivatives as Tubulin inhibitors
... molecular docking studies the compounds having electron withdrawing group shows good interaction with the beta-tubulin ...The Docking study shows Gln11, Asn101, Thr145 are important amino ... See full document
5
Membrane associated prostaglandin E synthase 1 is upregulated by proinflammatory cytokines in chondrocytes from patients with osteoarthritis
... several studies on the induction of COX-2 and its regula- tory mechanism in chondrocytes have already been pub- lished [16,36,37], this is the first report that mPGES-1, located downstream of COX-2, ... See full document
8
Quantitative estimation of new biologically active substances of derivated 4,5 dimethoxy N phenylanthranilic acids
... anthraniliс acids as to prospective class of biologically active substances which have various activities as that follow: analgetic, anti-inflammatory, fungistatic, diuretic, аnti-diuretic, ...of ... See full document
17
Synthesis, Characterization, Molecular Docking Studies and Antimicrobial Evaluation of N-Benzimidazol-1-Yl-Methyl-Benzamide Derivatives
... molecular docking studies were done and their inhibi- tory activity was tested against PDB ID: 1C14 micro- bial ...that N-(Benzimidazol-1-yl methyl)-benzamide derivatives act as potent ... See full document
8
Synthesis and molecular docking studies of 1 trityl 5 azaindazole derivatives
... All new compounds were subjected to molecular docking study with Murine double minutes-2(MDM2) receptor bind p53 and Pheripheral benzodiazepine receptor (PBR) cancer ...amino acids such as LEU43, ... See full document
20
Ascorbic acid enhances the inhibitory effect of aspirin on neuronal cyclooxygenase-2-mediated prostaglandin E2 production.
... is that ascorbic acid acts on the catalytic site of COX-2, which is the primary mechanism of action of aspirin-like drugs (Luong et al., 1996). Nevertheless, we excluded this possibility in the present study since ... See full document
6
INSILICO DESIGN AND MOLECULAR DOCKING STUDIES OF NOVEL 1, 2, 4- TRIAZOLE DERIVATIVES AS CYP-51 INHIBITORS
... modeling, docking is a method which predicts the preferred orientation of one molecule to a second when bound to each other to form a stable ...benzene derivatives. The objectives are to screen the 1,2,4- ... See full document
6
Molecular Docking Studies; Dietary Compounds As HIV 1 Protease Inhibitors
... ArgusLab: Arguslab is a freely available tool for various biological simultations. It was developed by Dr. Mark T Hompson and Planaria Software LLC. It is designed for windows platform. As the price of commercial ... See full document
76
Design, development, drug-likeness, and molecular docking studies of novel piperidin-4-imine derivatives as antitubercular agents
... general method for the synthesis of PB2–PB20 To an ethanolic solution of PB1 (2.29 g, 0.01 mol) with the appropriate amine (0.01 mol), sodium acetate (0.82 g, 0.01 mol) was added with stirring and it was refluxed for 3.5 ... See full document
25
Abstract
... further studies are needed to elucidate how COX−2 may be associated with genetic change in carcinogenesis in stomach that has not been clarified as well as in colon ... See full document
29
Cyclooxygenases, microsomal prostaglandin E synthase 1, and cardiovascular function
... and PGHS-2 KO mice on a mixed C57BL/6 × 129/Sv background. Thrombocytopenia was more pronounced (**P < 0.01) in PGHS-2–disrupted mice. Sudden death was induced more commonly (**P < 0.01) within 15 minutes of U46619 ... See full document
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